검색결과 : 7건
No. | Article |
---|---|
1 |
Design, synthesis, and characterization of a potent, nonpeptide, cell-permeable, bivalent smac mimetic that concurrently targets both the BIR2 and BIR3 domains in XIAP Sun HY, Nikolovska-Coleska Z, Lu JF, Meagher JL, Yang CY, Qiu S, Tomita Y, Ueda Y, Jiang S, Krajewski K, Roller PP, Stuckey JA, Wang SM Journal of the American Chemical Society, 129(49), 15279, 2007 |
2 |
Structure-based design of potent Grb2-SH2 domain antagonists not relying on phosphotyrosine mimics Jiang S, Li P, Peach ML, Bindu L, Worthy KW, Fisher RJ, Burke TR, Nicklaus M, Roller PP Biochemical and Biophysical Research Communications, 349(2), 497, 2006 |
3 |
Binding affinity difference induced by the stereochemistry of the sulfoxide bridge of the cyclic peptide inhibitors of Grb2-SH2 domain: NMR studies for the structural origin Shi YH, Song YL, Lin DH, Tan JZ, Roller PP, Li Q, Long YQ, Song GQ Biochemical and Biophysical Research Communications, 330(4), 1254, 2005 |
4 |
Structure-based design of potent non-peptide MDM2 inhibitors Ding K, Lu Y, Nikolovska-Coleska Z, Qiu S, Ding YS, Gao W, Stuckey J, Krajewski K, Roller PP, Tomita Y, Parrish DA, Deschamps JR, Wang SM Journal of the American Chemical Society, 127(29), 10130, 2005 |
5 |
Structure-based design of potent, conformationally constrained Smac mimetics Sun HY, Nikolovska-Coleska Z, Yang CY, Xu L, Liu ML, Tomita Y, Pan HG, Yoshioka Y, Krajewski K, Roller PP, Wang SM Journal of the American Chemical Society, 126(51), 16686, 2004 |
6 |
Potentiating effect of distant sites in non-phosphorylated cyclic peptide antagonists of the Grb2-SH2 domain Long YQ, Guo RB, Luo JH, Yang DJ, Roller PP Biochemical and Biophysical Research Communications, 310(2), 334, 2003 |
7 |
Structural basis for a non-phosphorus-containing cyclic peptide binding to Grb2-SH2 domain with high affinity Li P, Zhang MC, Peach ML, Zhang XD, Liu HP, Nicklaus M, Yang DJ, Roller PP Biochemical and Biophysical Research Communications, 307(4), 1038, 2003 |