검색결과 : 9건
| No. | Article |
|---|---|
| 1 |
Total Synthesis and Biological Evaluation of Tiancimycins A and B, Yangpumicin A, and Related Anthraquinone-Fused Enediyne Antitumor Antibiotics Nicolaou KC, Das D, Lu Y, Rout S, Pitsinos EN, Lyssikatos J, Schammel A, Sandoval J, Hammond M, Aujay M, Gavrilyuk J Journal of the American Chemical Society, 142(5), 2549, 2020 |
| 2 |
Synthesis and Biological Evaluation of Shishijimicin A-Type Linker-Drugs and Antibody-Drug Conjugates Nicolaou KC, Li RF, Chen QF, Lu ZY, Pitsinos EN, Schammel A, Lin BW, Gu C, Sarvaiya H, Tchelepi R, Valdiosera A, Clubb J, Barbour N, Sisodiya V, Sandoval J, Lee C, Aujay M, Gavrilyuk J Journal of the American Chemical Society, 142(29), 12890, 2020 |
| 3 |
Improved Total Synthesis of Tubulysins and Design, Synthesis, and Biological Evaluation of New Tubulysins with Highly Potent Cytotoxicities against Cancer Cells as Potential Payloads for Antibody-Drug Conjugates Nicolaou KC, Erande RD, Yin J, Vourloumis D, Aujay M, Sandoval J, Munneke S, Gavrilyuk J Journal of the American Chemical Society, 140(10), 3690, 2018 |
| 4 |
Streamlined Total Synthesis of Shishijimicin A and Its Application to the Design, Synthesis, and Biological Evaluation of Analogues thereof and Practical Syntheses of PhthNSSMe and Related Sulfenylating Reagents Nicolaou KC, Li RF, Lu ZY, Pitsinos EN, Alemany LB, Aujay M, Lee C, Sandoval J, Gavrilyuk J Journal of the American Chemical Society, 140(38), 12120, 2018 |
| 5 |
12,13-Aziridinyl Epothilones. Stereoselective Synthesis of Trisubstituted Olefinic Bonds from Methyl Ketones and Heteroaromatic Phosphonates and Design, Synthesis, and Biological Evaluation of Potent Antitumor Agents Nicolaou KC, Rhoades D, Wang YP, Bai RL, Hamel E, Aujay M, Sandoval J, Gavrilyuk J Journal of the American Chemical Society, 139(21), 7318, 2017 |
| 6 |
Streamlined Total Synthesis of Trioxacarcins and Its Application to the Design, Synthesis, and Biological Evaluation of Analogues Thereof. Discovery of Simpler Designed and Potent Trioxacarcin Analogues Nicolaou KC, Chen PX, Zhu SG, Cai Q, Erande RD, Li RF, Sun HB, Pulukuri KK, Rigol S, Aujay M, Sandoval J, Gavrilyuk J Journal of the American Chemical Society, 139(43), 15467, 2017 |
| 7 |
Total Synthesis and Biological Evaluation of Natural and Designed Tubulysins Nicolaou KC, Yun J, Mandal D, Erande RD, Klahn P, Jin M, Aujay M, Sandoval J, Gavrilyuk J, Vourloumis D Journal of the American Chemical Society, 138(5), 1698, 2016 |
| 8 |
Synthesis and Biological Investigation of Delta(12)-Prostaglandin J3 (Delta(12)-PGJ(3)) Analogues and Related Compounds Nicolaou KC, Pulukuri KK, Rigol S, Heretsch P, Yu RC, Grove CI, Hale CRH, ElMarrouni A, Fetz V, Bronstrup M, Aujay M, Sandoval J, Gavrilyuk J Journal of the American Chemical Society, 138(20), 6550, 2016 |
| 9 |
Tyrosine Bioconjugation through Aqueous Ene-Type Reactions: A Click-Like Reaction for Tyrosine Ban H, Gavrilyuk J, Barbas CF Journal of the American Chemical Society, 132(5), 1523, 2010 |